{"id":2918,"date":"2016-06-15T16:15:57","date_gmt":"2016-06-15T19:15:57","guid":{"rendered":"https:\/\/prodoctor.net\/blog\/?p=2918"},"modified":"2021-06-10T16:40:52","modified_gmt":"2021-06-10T19:40:52","slug":"pesquisadores-descobrem-remedios-para-antigas-doencas","status":"publish","type":"post","link":"https:\/\/prodoctor.net\/blog\/pesquisadores-descobrem-remedios-para-antigas-doencas\/","title":{"rendered":"Pesquisadores descobrem rem\u00e9dios para antigas doen\u00e7as"},"content":{"rendered":"<p>Antigas doen\u00e7as, cujo combate n\u00e3o tem merecido a devida aten\u00e7\u00e3o atrav\u00e9s de campanhas pela&nbsp;Organiza\u00e7\u00e3o Mundial da Sa\u00fade (OMS), come\u00e7am a ser <strong>vistas por um prisma diferente<\/strong>. E a&nbsp;iniciativa para lutar contra algumas delas, como o Mal de Chagas e a Leishmaniose, <strong>j\u00e1 apresenta&nbsp;resultados<\/strong>, como as <strong>drogas formuladas por pesquisadores do Brasil<\/strong>. A expectativa dos estudiosos&nbsp;reside no fato de que existe a possibilidade de serem desenvolvidas <strong>mol\u00e9culas com novas&nbsp;formula\u00e7\u00f5es farmac\u00eauticas<\/strong>, associa\u00e7\u00e3o de drogas e tamb\u00e9m em formas <strong>menos t\u00f3xicas<\/strong> para&nbsp;aplica\u00e7\u00e3o dos rem\u00e9dios dispon\u00edveis no mercado.&nbsp;<\/p>\n<p>Causada pelo protozo\u00e1rio Trypanosoma cruzi, <strong>a Doen\u00e7a (Mal) de Chagas<\/strong> \u00e9 transmitida pelo inseto&nbsp;barbeiro, atingindo 8 milh\u00f5es de pessoas em todo o planeta, e provocando a morte de 12 mil a cada&nbsp;ano, conforme dados da OMS. J\u00e1 a <strong>Leishmaniose<\/strong> \u00e9 transmitida por insetos hemat\u00f3fagos conhecidos&nbsp;(fleb\u00f3tomos ou flebotom\u00edneos), com duas formas de manifesta\u00e7\u00e3o: a visceral, que pode matar, e a&nbsp;cut\u00e2nea. Segundo a Organiza\u00e7\u00e3o Mundial da Sa\u00fade, cerca de 12 milh\u00f5es de pessoas podem estar&nbsp;infectadas, constatando-se anualmente a morte de 30 mil pessoas.<\/p>\n<p>Os pesquisadores Wagner Vilegas, do Instituto de Bioci\u00eancias da Universidade Estadual Paulista&nbsp;(Unesp), em S\u00e3o Vicente (SP), Emerson Ferreira Queiroz, da Universidade de Genebra, na Su\u00ed\u00e7a, e&nbsp;Cl\u00e1udia Quintino da Rocha, da Universidade Federal do Maranh\u00e3o (UFMA), isolaram <strong>uma nova&nbsp;fam\u00edlia de mol\u00e9culas<\/strong> a partir da planta <strong>Arrabidaea brachypoda<\/strong>, conhecida no cerrado brasileiro&nbsp;como cervejinha-do-campo e <strong>usada contra c\u00e1lculos renais<\/strong>. A partir dos resultados de pesquisas <em>in&nbsp;vitro<\/em> e <em>in vivo<\/em>, com animais de laborat\u00f3rio, avaliaram que uma mol\u00e9cula da fam\u00edlia tem potencial&nbsp;para o <strong>desenvolvimento de um novo medicamento<\/strong>.&nbsp;<\/p>\n<p>Nas doses testadas, a subst\u00e2ncia n\u00e3o apresentou toxicidade, proporcionando um alento&nbsp;na luta contra o Mal de Chagas. O&nbsp;benznidazol, droga mais usada&nbsp;hoje no Brasil, provoca fortes efeitos colaterais, com rea\u00e7\u00f5es al\u00e9rgicas cut\u00e2neas, enjoos e v\u00f4mitos.&nbsp;A pesquisa caminha para seu est\u00e1gio final, <strong>quando se espera comprovar sua efic\u00e1cia<\/strong>, devendo&nbsp;ent\u00e3o ser intensificada a busca por <strong>parceiros na ind\u00fastria farmac\u00eautica<\/strong> para viabilizar os testes&nbsp;cl\u00ednicos em seres humanos.&nbsp;<\/p>\n<p>Enquanto isso, no Instituto Adolfo Lutz, o pesquisador Andr\u00e9 Tempone trabalha&nbsp;com equipes multidisciplinares <strong>abrangendo o reposicionamento de f\u00e1rmacos<\/strong> j\u00e1 existentes e&nbsp;<strong>associa\u00e7\u00f5es terap\u00eauticas<\/strong>. Est\u00e1 em<strong> estudos&nbsp;o potencial terap\u00eautico<\/strong> de antidepressivos orais com&nbsp;base na sertralina para a Leishmaniose Visceral e Cut\u00e2nea e para o Mal de Chagas.&nbsp;Os testes com animais est\u00e3o sendo realizados pelo Instituto, pelas universidades de Dundee&nbsp;(Esc\u00f3cia), San Pablo (Espanha) e na Faculdade de Ci\u00eancias Farmac\u00eauticas da Universidade de S\u00e3o&nbsp;Paulo (FCF-USP), com o apoio da FAPESP. Em caso de resultados positivos, o passo seguinte ser\u00e1&nbsp;usar a sertralina com o benznidazol para combater a doen\u00e7a.<\/p>\n<h4>Associa\u00e7\u00e3o de drogas<\/h4>\n<p>Para<strong> enfrentar a&nbsp;Leishmaniose<\/strong>, os testes com a sertralina ser\u00e3o feitos&nbsp;em associa\u00e7\u00e3o com as drogas anfotericina&nbsp;B e miltefosina. Importante destacar que essa segunda droga<strong> ainda \u00e9 alvo de estudos<\/strong> cl\u00ednicos no&nbsp;Brasil, onde <strong>o medicamento mais utilizado<\/strong> para <strong>combater a doen\u00e7a \u00e9 um composto com antim\u00f4nio<\/strong>.&nbsp;O pesquisador ressalta que o antim\u00f4nio trata o paciente, mas <strong>n\u00e3o elimina 100% o parasita<\/strong>, al\u00e9m de&nbsp;provocar <strong>efeitos colaterais<\/strong> adversos graves, principalmente para doentes card\u00edacos e renais.<\/p>\n<p>J\u00e1 a pesquisadora Bartira Rossi-Bergmann, da Universidade Federal do Rio de Janeiro (UFRJ)<strong>&nbsp;concentra seus estudos na luta contra a Leishmaniose Cut\u00e2nea<\/strong>, que, embora n\u00e3o seja letal, deixa um&nbsp;rastro de graves consequ\u00eancias sociais para <strong>1,2 milh\u00e3o de infectados<\/strong> por ano em todo o planeta. Em&nbsp;vez das inje\u00e7\u00f5es di\u00e1rias de antim\u00f4nio, seu trabalho prev\u00ea a <strong>aplica\u00e7\u00e3o de um medicamento em dose&nbsp;\u00fanica,<\/strong>&nbsp;implantando nanopart\u00edculas no local infectado, com a libera\u00e7\u00e3o gradual da droga na&nbsp;pele.<\/p>\n<p>Tamb\u00e9m est\u00e3o em estudos<strong> duas possibilidades de drogas<\/strong> que poder\u00e3o ser conjugadas em um \u00fanico implante.&nbsp;A primeira, e mais promissora, utiliza a s\u00edntese de uma mol\u00e9cula identificada da <strong>planta&nbsp;Piper&nbsp;aduncum<\/strong>, da fam\u00edlia das pimentas, que ter\u00e1 que passar por testes em animais e seres humanos. J\u00e1 a&nbsp;segunda, com a utiliza\u00e7\u00e3o da <strong>anfotericina B<\/strong>, j\u00e1 usada no tratamento da Leishmaniose. Conforme a&nbsp;pesquisadora, testes realizados com camundongos indicam que o implante da anfotericina B na pele&nbsp;n\u00e3o gera os efeitos colaterais comuns ao medicamento, quando a droga \u00e9 injetada no m\u00fasculo.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Antigas doen\u00e7as, cujo combate n\u00e3o tem merecido a devida aten\u00e7\u00e3o atrav\u00e9s de campanhas pela&nbsp;Organiza\u00e7\u00e3o Mundial da Sa\u00fade (OMS), come\u00e7am&#8230;<\/p>\n","protected":false},"author":1,"featured_media":19567,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"_kad_blocks_custom_css":"","_kad_blocks_head_custom_js":"","_kad_blocks_body_custom_js":"","_kad_blocks_footer_custom_js":"","_kadence_starter_templates_imported_post":false,"_kad_post_transparent":"","_kad_post_title":"","_kad_post_layout":"","_kad_post_sidebar_id":"","_kad_post_content_style":"","_kad_post_vertical_padding":"","_kad_post_feature":"","_kad_post_feature_position":"","_kad_post_header":false,"_kad_post_footer":false,"footnotes":""},"categories":[415,413],"tags":[],"class_list":["post-2918","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-medicamentos-e-farmacia","category-medicina-e-saude"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.0 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Pesquisadores 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